又称:DSPE-PCB;聚甜菜碱甲基水性聚氨酯酯-磷脂;男女性甜菜碱缩聚物胶束(DSPE-PCB)
描素:的使用两性之间甜菜碱缩聚物胶束(DSPE-PCB)来模仿衣壳木马病毒的表面上特殊性(图1a),并封裝模板血清。聚羧爽口莱碱(PCB)确认质子帮助蛋清质装运蛋清1(PAT1)吸收上皮细胞膜层(图1b)。PAT1能有助于甜菜碱和甜菜碱衍化物渗透性到上皮人体细胞层。
Because of the sharp contrast in polarity between the superhydrophilic tail and the superhydrophobic head of DSPE–PCB 5K, its micelles stabilize docetaxel at extremely dilute conditions, at which conventional micelles dissociate. In vivo, the ultrastability of the formulation enables a larger amount of drug to reach the tumour through the enhanced permeability and retention effect. Chemical structure reproduced from ref. 8, Macmillan Publishers Ltd.
定制产品:
DSPE-PEG-cRGD 磷脂-聚乙二醇-靶向穿膜肽CRGD
DSPE-PEG-RGD 磷脂-聚乙二醇-靶向穿膜肽RGD
DSPE-PEG-iRGD 磷脂-聚乙二醇-靶向穿膜肽IRGD
DSPE-PEG-R6H4 磷脂-聚乙二醇-PH响应性穿膜肽R6H4
DSPE-PEG-MPG 磷脂-聚乙二醇-PH响应性穿膜肽MPG
DSPE-PEG-SEARYL-R8 磷脂-聚乙二醇-PH响应性穿膜肽SEARYL-R8
DSPE-PEG-EB1 磷脂-聚乙二醇-PH响应性穿膜肽EB1
DSPE-PEG-PF6 磷脂-聚乙二醇-PH响应性穿膜肽PF6
DSPE-PEG-TAT 磷脂-聚乙二醇-靶向穿膜肽TAT
DSPE-PEG-R8 磷脂-聚乙二醇-靶向穿膜肽R8
DSPE-PEG-Angiopep 磷脂-聚乙二醇-*微环境穿膜肽
DSPE-PEG-GE11 磷脂-聚乙二醇-*细胞表皮生长因子肽GE11
DSPE-PEG-TH 磷脂-聚乙二醇-PH响应性穿膜肽TH
DSPE-PEG-APRPG 磷脂-聚乙二醇-*新生靶向肽APRPG
DSPE-PEG-NGR 磷脂-聚乙二醇-*新生靶向肽NRG
DSPE-PEG-PSHB 磷脂-聚乙二醇-卵泡刺*多肽PSHB
DSPE-PEG-NYZL1 磷脂-聚乙二醇-膀胱*靶向肽NYZL1
DSPE-PEG-HAIYPRH 磷脂-聚乙二醇-转铁蛋白靶向肽HAIYPRH
DSPE-PEG-SP94 磷脂-聚乙二醇-肝*特异靶向肽SP94
DSPE-PEG-PTP 磷脂-聚乙二醇-**靶向肽PTP
DSPE-PEG-VIP 磷脂-聚乙二醇-活性肠肽VIP
DSPE-PEG-OTC 磷脂-聚乙二醇-奥曲肽
CPP-PEG-DSPE 细胞穿透肽靶向肽修饰脂质体